Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Kappa-type opioid receptor' and Ligand = 'BDBM50084275'
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50084275(7,7-Spiro analogue ofBuprinorphine | CHEMBL31605)
Affinity DataKi:  1.30nMAssay Description:Binding affinity to cloned human Opioid receptor kappa 1 transfected into hamster ovary cells using [3H]U-69593 as a radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of Bristol

Curated by ChEMBL
LigandPNGBDBM50084275(7,7-Spiro analogue ofBuprinorphine | CHEMBL31605)
Affinity DataEC50:  1.60nMAssay Description:GTPgammaS binding in cloned human Opioid receptor kappa 1 transfected into hamster ovary cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed