Affinity DataKi: 0.0520nMAssay Description:Displacement of radioligand from human KISS1R transfected in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Agonist activity at rat KISS1R transfected in CHO cells assessed as intracellular calcium flux after 24 hrs by functional FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.80nMAssay Description:Agonist activity at human KISS1R transfected in CHO cells assessed as intracellular calcium flux after 24 hrs by functional FLIPR assayMore data for this Ligand-Target Pair