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Found 2 Enz. Inhib. hit(s) with Target = 'KiSS-1 receptor' and Ligand = 'BDBM50320802'
TargetKiSS-1 receptor(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50320802(CHEMBL1164939 | N-[4-{3-[(4-Aminobutanoyl)amino]ph...)
Affinity DataIC50:  34nMAssay Description:Displacement of [125I]metastin(40-54) from human GPR54 receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
Takeda Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50320802(CHEMBL1164939 | N-[4-{3-[(4-Aminobutanoyl)amino]ph...)
Affinity DataIC50:  1.40E+3nMAssay Description:Antagonist activity at human GPR54 receptor expressed in CHO cells assessed as inhibition of metastin(40-54)-induced intracellular calcium mobilizati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed