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Found
1
Enz. Inhib. hit(s) with Target = 'MLL1-WRAD2 complex' and Ligand = 'BDBM552980'
Target
MLL1-WRAD2 complex
(Homo sapiens (Human))
Propellon Therapeutics
US Patent
Ligand
BDBM552980
(N-[4-fluoro-2-(4- methylpiperazin-1-yl)-5- [6-(oxa...)
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Affinity Data
IC50: 1.00E+3nM
Assay Description:
Compound potency was assessed through incorporation of 3H-SAM into oligonucleosomes purified from HeLa cells. Specifically, recombinant human MLL1 (a...
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Target Info
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Ligand Info
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US Patent
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