Found 6 Enz. Inhib. hit(s) with Target = 'Mas-related G-protein coupled receptor member X1' and Ligand = 'BDBM224021'
TargetMas-related G-protein coupled receptor member X1(Homo sapiens (Human))
Johns Hopkins University
Curated by ChEMBL
Johns Hopkins University
Curated by ChEMBL
Affinity DataEC50: 50nMAssay Description:Agonist activity at human MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
TargetMas-related G-protein coupled receptor member X1(Rattus norvegicus)
Johns Hopkins University
Curated by ChEMBL
Johns Hopkins University
Curated by ChEMBL
Affinity DataEC50: 316nMAssay Description:Agonist activity at rat MrgX1 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair
TargetMas-related G-protein coupled receptor member X1(Homo sapiens (Human))
Johns Hopkins University
Curated by ChEMBL
Johns Hopkins University
Curated by ChEMBL
Affinity DataEC50: 50nMAssay Description:Agonist activity at human MrgprX1More data for this Ligand-Target Pair
Affinity DataEC50: 300nMAssay Description:Agonist activity at mouse MRGPRC11More data for this Ligand-Target Pair
TargetMas-related G-protein coupled receptor member X1(Rattus norvegicus)
Johns Hopkins University
Curated by ChEMBL
Johns Hopkins University
Curated by ChEMBL
Affinity DataEC50: 300nMAssay Description:Agonist activity at rat MRGPRCMore data for this Ligand-Target Pair
Affinity DataEC50: 251nMAssay Description:Agonist activity at mouse MrgC11 transfected in HEK293 cells by FLIPR assayMore data for this Ligand-Target Pair