Affinity DataIC50: 7.30E+3nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]-hAGRP(82-132)More data for this Ligand-Target Pair
Affinity DataIC50: 1.03E+4nMAssay Description:Inhibitory concentration towards melanocortin MC4 receptor by displacing radioligand [125I]NDP-MSHMore data for this Ligand-Target Pair
Affinity DataEC50: 1.59E+4nMAssay Description:Effective concentration against mouse melanocortin MC4 receptor; Partial agonistMore data for this Ligand-Target Pair