Affinity DataIC50: 0.0900nMAssay Description:Binding affinity against human Melanocortin 5 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.900nMAssay Description:Displacement of [125I][Nle4,Dphe7]-alpha-MSH from human MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.20nMAssay Description:Agonist activity at human MC5R expressed in HEK293 cells assessed as stimulation of intracellular cAMP levelMore data for this Ligand-Target Pair
Affinity DataEC50: 0.120nMAssay Description:Binding affinity against human Melanocortin 5 receptorMore data for this Ligand-Target Pair