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Found 2 Enz. Inhib. hit(s) with Target = 'Melanocortin receptor 5' and Ligand = 'BDBM50268799'
TargetMelanocortin receptor 5(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50268799(Ac-Nle-c[Asp-His-DNal(2')-trans-4-guanidinyl-Pro-T...)
Affinity DataIC50:  22nMAssay Description:Displacement of [125I][Nle4,Dphe7]-alpha-MSH from human MC5R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50268799(Ac-Nle-c[Asp-His-DNal(2')-trans-4-guanidinyl-Pro-T...)
Affinity DataEC50:  2.40E+3nMAssay Description:Agonist activity at human MC5R expressed in HEK293 cells assessed as stimulation of intracellular cAMP levelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed