Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Melanocyte-stimulating hormone receptor' and Ligand = 'BDBM250638'
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Palatin Technologies

US Patent
LigandPNGBDBM250638(US9447148, 9.6)
Affinity DataKi:  0.0700nM ΔG°:  -60.3kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay was performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMCR-1a or hMCR-...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Palatin Technologies

US Patent
LigandPNGBDBM250638(US9447148, 9.6)
Affinity DataEC50:  0.0140nMpH: 7.5 T: 2°CAssay Description:Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent