Found 6 Enz. Inhib. hit(s) with Target = 'Melanocyte-stimulating hormone receptor' and Ligand = 'BDBM50121885'
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Roche Research Center
Curated by ChEMBL
Roche Research Center
Curated by ChEMBL
Affinity DataIC50: 580nMAssay Description:Binding affinity towards human melanocortin receptor hMC4R by using radioligand NDP-MSH; not determinedMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Roche Research Center
Curated by ChEMBL
Roche Research Center
Curated by ChEMBL
Affinity DataIC50: 580nMAssay Description:Binding affinity towards human Melanocortin 1 receptor using radiolabeled NDP-MSH displacementMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Roche Research Center
Curated by ChEMBL
Roche Research Center
Curated by ChEMBL
Affinity DataEC50: 10nMAssay Description:Agonist activity in HEK293 cells transfected with human MC1R by cAMP accumulationMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Roche Research Center
Curated by ChEMBL
Roche Research Center
Curated by ChEMBL
Affinity DataEC50: 10nMAssay Description:Agonist activity against human melanocortin receptor hMC1RMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Roche Research Center
Curated by ChEMBL
Roche Research Center
Curated by ChEMBL
Affinity DataEC50: 10nMAssay Description:Agonist activity against human melanocortin receptor hMC1R at 50% maximum cAMP accumulationMore data for this Ligand-Target Pair
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Roche Research Center
Curated by ChEMBL
Roche Research Center
Curated by ChEMBL
Affinity DataEC50: 10nMAssay Description:Effective concentration required for cAMP accumulation mediated by human Melanocortin 1 receptor in HEK293 cellsMore data for this Ligand-Target Pair