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Found 2 Enz. Inhib. hit(s) with Target = 'Melatonin receptor type 1A/1B' and Ligand = 'BDBM50037242'
TargetMelatonin receptor type 1A/1B(Homo sapiens (Human))
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandPNGBDBM50037242(CHEMBL323332 | N-(2-(5-methoxybenzofuran-3-yl)ethy...)
Affinity DataIC50:  1.70nMAssay Description:Monophasic inhibitory concentration against melatonin receptor was measured on ovine pars tuberalis membrane.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A/1B(Homo sapiens (Human))
Institut De Chimie Pharmaceutique

Curated by ChEMBL
LigandPNGBDBM50037242(CHEMBL323332 | N-(2-(5-methoxybenzofuran-3-yl)ethy...)
Affinity DataKd:  0.859nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed