Found 2 Enz. Inhib. hit(s) with Target = 'Melatonin receptor type 1A/1B' and Ligand = 'BDBM50037242'
TargetMelatonin receptor type 1A/1B(Homo sapiens (Human))
Institut De Chimie Pharmaceutique
Curated by ChEMBL
Institut De Chimie Pharmaceutique
Curated by ChEMBL
Affinity DataIC50: 1.70nMAssay Description:Monophasic inhibitory concentration against melatonin receptor was measured on ovine pars tuberalis membrane.More data for this Ligand-Target Pair
TargetMelatonin receptor type 1A/1B(Homo sapiens (Human))
Institut De Chimie Pharmaceutique
Curated by ChEMBL
Institut De Chimie Pharmaceutique
Curated by ChEMBL
Affinity DataKd: 0.859nMAssay Description:Binding affinity to melatonin receptor measured on ovine pars tuberalis membraneMore data for this Ligand-Target Pair