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Report error Found 2 Enz. Inhib. hit(s) with Target = 'Metabotropic glutama...
TargetMetabotropic glutamate receptor 1(RAT)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50224403(8-(4-methylphenyl)-1H-pyrazolo[3'',4'':4',5']pyrid...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]9-Dimethylamino-3-(4-methoxy-phenyl)-3H-pyrido[3',2':4,5]thieno[3,2-d]pyrimidin-4-one from mGluR1 in rat cerebellum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50224403(8-(4-methylphenyl)-1H-pyrazolo[3'',4'':4',5']pyrid...)
Affinity DataIC50:  17nMAssay Description:Antagonist activity at human mGluR1a expressed in CHO cells assessed by measuring intracellular calcium by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed