TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Displacement of [3H]-DAMGO from mu opioid receptor (unknown origin) expressed in CHO cells at 10 uMMore data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 7.20nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 1.10E+4nMAssay Description:Agonist activity at human MOR receptor expressed in HTLA cells co-expressing TEV-fused-beta-arrestin2 assessed as induction of beta-arrestin2 recruit...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 7.30nMAssay Description:Agonist activity at human MOR expressed in HEK293T cells assessed as inhibition of forskolin-stimulated cAMP accumulation incubated for 30 mins by Gl...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
University Of Health Sciences & Pharmacy At St. Louis
Curated by ChEMBL
Affinity DataEC50: 1.10E+4nMAssay Description:Agonist activity at human MOR receptor expressed in HTLA cells co-expressing TEV-fused-beta-arrestin2 assessed as induction of beta-arrestin2 recruit...More data for this Ligand-Target Pair