Found 17 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1' and Ligand = 'BDBM50004665'
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Arizona
Curated by PDSP Ki Database
University Of Arizona
Curated by PDSP Ki Database
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Arizona
Curated by PDSP Ki Database
University Of Arizona
Curated by PDSP Ki Database
Affinity DataKi: 1.10nMAssay Description:Binding affinity to human cloned muscarinic M1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Arizona
Curated by PDSP Ki Database
University Of Arizona
Curated by PDSP Ki Database
Affinity DataKi: 17nMAssay Description:Inhibition of [3H]- oxotremorine-M binding to human Muscarinic acetylcholine receptor M1 expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:Binding affinity at [3H]PZ radiolabeled muscarinic M1 receptor in rat cortex.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 196nMAssay Description:Compound was evaluated for its binding affinity towards muscarinic acetylcholine receptor in rat cortexMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
TargetMuscarinic acetylcholine receptor M1(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataKi: 630nMAssay Description:Binding affinity to Muscarinic acetylcholine receptor M1 by measuring its ability to displace [3H]pirenzepine from rat cerebral cortexMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Arizona
Curated by PDSP Ki Database
University Of Arizona
Curated by PDSP Ki Database
Affinity DataIC50: 2.30nMAssay Description:Ability to displace [3H]-oxotremorine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Binding affinity against Muscarinic receptor M1 in rat brain using [3H]-PZ (pirenzepine) radioligand at a concentration of 1 nMMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataIC50: 113nMAssay Description:Ability to displace [3H]-pirenzepine (pir) from muscarinic acetylcholine receptor M1 in rat cortical tissue.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Medical Research Division Of American Cyanamid
Curated by ChEMBL
Affinity DataIC50: 360nMAssay Description:Compound was evaluated for the displacement of the muscarinic QNB in a genetically transformed rat cell line (m1c2) transfected with cloned m1 recept...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Arizona
Curated by PDSP Ki Database
University Of Arizona
Curated by PDSP Ki Database
Affinity DataIC50: 364nMAssay Description:Displacement of [3H]-QNB in genetically transformed mouse cell line (m1C2) transfected with Muscarinic acetylcholine receptor M1More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Arizona
Curated by PDSP Ki Database
University Of Arizona
Curated by PDSP Ki Database
Affinity DataIC50: 9.00E+3nMAssay Description:Compound was evaluated for its ability to displace [3H]-N-methylscopolamine ([3H]-NMS) binding to cloned CHO cell lines expressing Muscarinic acetylc...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Arizona
Curated by PDSP Ki Database
University Of Arizona
Curated by PDSP Ki Database
Affinity DataIC50: 2.71E+4nMAssay Description:Ability to displace [3H]-N-methylscopolamine from Muscarinic acetylcholine receptor M1 expressed in CHO cells.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Arizona
Curated by PDSP Ki Database
University Of Arizona
Curated by PDSP Ki Database
Affinity DataEC50: 390nMAssay Description:In Vitro evaluation of the compound activity at the cloned Human Muscarinic acetylcholine receptor M1 determined by receptor selection and amplificat...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
University Of Arizona
Curated by PDSP Ki Database
University Of Arizona
Curated by PDSP Ki Database
Affinity DataEC50: 1.60nMAssay Description:Agonist activity at human m1 muscarinic acetylcholine receptor expressed in HEK293 cells assessed as calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
Affinity DataEC50: 270nMAssay Description:Tested against Muscarinic acetylcholine receptor M1 expressed in A9 L cell lineMore data for this Ligand-Target Pair