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Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M2' and Ligand = 'BDBM50326219'
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50326219(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
Affinity DataKi:  980nMAssay Description:Agonist activity at human muscarinic M2 receptor expressed in CHO-K1 cells coexpressing Galpha16 subunit assessed as increase of acetylcholine-induce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50326219(4-(4-butylpiperidin-1-yl)-1-o-tolylbutan-1-one | C...)
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity to human muscarinic M2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed