Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M2' and Ligand = 'BDBM50366775'
Affinity DataKi: 2.60nMAssay Description:Affinity for rat M1 acetylcholine receptor using [3H]-AF DX 384 displacement.More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Pipeline Therapeutics
Curated by ChEMBL
Pipeline Therapeutics
Curated by ChEMBL
Affinity DataIC50: 63nMAssay Description:Antagonist activity at human recombinant muscarinic receptor M2 expressed in CHO-K1 cells assessed as EC80 acetylcholine-induced calcium flux incubat...More data for this Ligand-Target Pair