Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with Target = 'Na(+)/H(+) exchange regulatory cofactor NHE-RF1 [133-300]' and Ligand = 'BDBM228839'
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1 [133-300](Human)
The University of Queensland

LigandPNGBDBM228839(biotin-DEEASCPERPPALLQEEWETVM | b-PTHRct-22)
Affinity DataKi:  7.00E+3nM ΔG°:  -29.2kJ/molepH: 7.4 T: 2°CAssay Description:Competition assays were performed in FP buffer (DTT was avoided for Cys-PTHRct-9) containing fixed concentrations of both the fluorescently labeled p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2017
Entry Details Article
PubMed
TargetNa(+)/H(+) exchange regulatory cofactor NHE-RF1 [133-300](Human)
The University of Queensland

LigandPNGBDBM228839(biotin-DEEASCPERPPALLQEEWETVM | b-PTHRct-22)
Affinity DataKd:  1.15E+4nMpH: 7.4 T: 2°CAssay Description:SPR measurements were performed with a Biacore X100 instrument (GE Healthcare Life Sciences, Piscataway, NJ) at 15.0 °C. The biotinylated PTHRct-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2017
Entry Details Article
PubMed