Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor subunit alpha-3/beta-4' and Ligand = 'BDBM50498762'
LigandPNGBDBM50498762(CHEMBL3622601)
Affinity DataEC50: <1.00E+6nMAssay Description:Agonist activity at rat neuronal acetylcholine receptor subunit alpha3beta4 expressed in HEK293 cells at 1 mM by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50498762(CHEMBL3622601)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at rat neuronal acetylcholine receptor subunit alpha3beta4 expressed in HEK293 cells at 1 mM by FMP assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50498762(CHEMBL3622601)
Affinity DataKi:  1.00E+5nMAssay Description:Displacement of [3H]epibatidine from rat neuronal acetylcholine receptor subunit alpha3beta4 expressed in HEK293 cell membranes incubated for 4 hrs b...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
LigandPNGBDBM50498762(CHEMBL3622601)
Affinity DataKi:  1.00E+5nMAssay Description:Displacement of [3H]epibatidine from rat neuronal acetylcholine receptor subunit alpha3beta4 expressed in HEK293 cell membranes incubated for 4 hrs b...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed