Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor subunit alpha-3' and Ligand = 'BDBM50275265'
TargetNeuronal acetylcholine receptor subunit alpha-3(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50275265(3-((Azetidine-1-carbonyloxy)-1-methylpropyl)dimeth...)
Affinity DataEC50: >3.16E+5nMAssay Description:Agonist activity at human alpha-3-beta-4 nAChR expressed in Xenopus oocytes by two-electrode voltage clamp techniqueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Rat)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50275265(3-((Azetidine-1-carbonyloxy)-1-methylpropyl)dimeth...)
Affinity DataKi:  23nMAssay Description:Agonist activity at rat alpha-3-beta-4 nAChR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Rat)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50275265(3-((Azetidine-1-carbonyloxy)-1-methylpropyl)dimeth...)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [3H]epibatidine from rat recombinant alpha-3-beta-4 nAChR expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/19/2012
Entry Details Article
PubMed