Report error Found 8 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor subunit alpha-4/beta-2' and Ligand = 'BDBM50143314'
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
University of Milan
Curated by ChEMBL
University of Milan
Curated by ChEMBL
Affinity DataKd: 0.0300nMAssay Description:Binding affinity to alpha4beta2 nACh receptor (unknown origin) expressed in Xenopus oocytesMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Sassari
Curated by ChEMBL
University of Sassari
Curated by ChEMBL
Affinity DataKi: 0nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR in rat cerebral cortex membraneMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Sassari
Curated by ChEMBL
University of Sassari
Curated by ChEMBL
Affinity DataKi: 0.0180nMAssay Description:Inhibition of [3H]epibatidine binding at the nicotinic acetylcholine receptor alpha4-beta2 in male rat cerebral cortexMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Sassari
Curated by ChEMBL
University of Sassari
Curated by ChEMBL
Affinity DataKi: 0.0260nMAssay Description:Inhibition of [3H]epibatidine binding to Nicotinic acetylcholine receptor alpha4-beta2 from rat membranes from ref 16More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Sassari
Curated by ChEMBL
University of Sassari
Curated by ChEMBL
Affinity DataKi: 0.0550nMAssay Description:Inhibition of [3H]nicotine binding to Nicotinic acetylcholine receptor alpha4-beta2 from rat membranes from ref 15More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Sassari
Curated by ChEMBL
University of Sassari
Curated by ChEMBL
Affinity DataKi: 0.0580nMAssay Description:Non-specific binding in presence of 300 uM nicotine at nicotinic acetylcholine receptor alpha4-beta2 in rat cerebral cortex membranesMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Sassari
Curated by ChEMBL
University of Sassari
Curated by ChEMBL
Affinity DataKi: 0.0580nMAssay Description:Inhibition of [3H]nicotine binding to Nicotinic acetylcholine receptor alpha4-beta2 from rat membranes from ref 14More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
University of Sassari
Curated by ChEMBL
University of Sassari
Curated by ChEMBL
Affinity DataKi: 0.260nMAssay Description:Inhibition of [3H]nicotine binding to Nicotinic acetylcholine receptor alpha4-beta2 from rat membranesMore data for this Ligand-Target Pair
