Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with Target = 'Neuronal acetylcholine receptor subunit alpha-4/beta-2' and Ligand = 'BDBM50246826'
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50246826BDBM50246826(CHEMBL4084577)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at rat alpha4beta2 nAChR expressed in HEK cells assessed as inhibition of epibatidine-induced membrane potential preincubated for...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2019
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Rat)
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50246826BDBM50246826(CHEMBL4084577)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]epibatidine from rat alpha4beta2 nAChR expressed in HEK cell membranes after 2 hrsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2019
Entry Details Article
PubMed