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Found 5 Enz. Inhib. hit(s) with Target = 'Neurotensin receptor type 1' and Ligand = 'BDBM50509513'
TargetNeurotensin receptor type 1(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50509513(CHEMBL4537266)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H] UR-MK300 from human neurotensin receptor 1 stably expressed in CHO cells incubated in dark after 30 mins by liquid scintillation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50509513(CHEMBL4537266)
Affinity DataKi:  2nMAssay Description:Displacement of [3H] UR-MK300 from human neurotensin receptor 1 expressed in HT-29 cells incubated in dark after 30 mins by liquid scintillation coun...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50509513(CHEMBL4537266)
Affinity DataKd:  26nMAssay Description:Binding affinity to human neurotensin receptor 1 stably expressed in CHO cells incubated for 60 mins in presence of NT (8 to 13) without compound was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50509513(CHEMBL4537266)
Affinity DataKd:  6.80nMAssay Description:Binding affinity to human neurotensin receptor 1 stably expressed in CHO cells incubated for 75 mins in presence of NT (8 to 13) followed by compound...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNeurotensin receptor type 1(Homo sapiens (Human))
University of Regensburg

Curated by ChEMBL
LigandPNGBDBM50509513(CHEMBL4537266)
Affinity DataEC50:  0.372nMAssay Description:Agonist activity at human neurotensin receptor 1 expressed in CHO cells assessed as increase in intracellular calcium by Fluo-4 dye based fluorescenc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed