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Found 8 Enz. Inhib. hit(s) with Target = 'Nischarin' and Ligand = 'BDBM50138500'
TargetNischarin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50138500(2-((E)-Styryl)-4,5-dihydro-1H-imidazole | 2-styryl...)
Affinity DataKi:  2nMAssay Description:Binding affinity for imidazoline receptor I-2 in rabbit kidney homogenate (relative to [3H]-Idazoxan radioligand)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50138500(2-((E)-Styryl)-4,5-dihydro-1H-imidazole | 2-styryl...)
Affinity DataKi:  10nMAssay Description:Binding affinity for rat imidazoline receptor I-1 from crude P2 membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)TBA
LigandPNGBDBM50138500(2-((E)-Styryl)-4,5-dihydro-1H-imidazole | 2-styryl...)
Affinity DataKi:  19nMAssay Description:Binding affinity to I1 imidazoline binding site in Rattus norvegicus (rat) PC12 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNischarin(RAT)TBA
LigandPNGBDBM50138500(2-((E)-Styryl)-4,5-dihydro-1H-imidazole | 2-styryl...)
Affinity DataKi:  19nMAssay Description:Displacement of [125I]-p-iodoclonidine from I1 receptor imidazoline binding site in rat PC12 cell membranes after 30 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)TBA
LigandPNGBDBM50138500(2-((E)-Styryl)-4,5-dihydro-1H-imidazole | 2-styryl...)
Affinity DataKi:  19nMAssay Description:Displacement of [125I]PIC from Imidazoline-1 receptor in rat PC12 cell membrane by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50138500(2-((E)-Styryl)-4,5-dihydro-1H-imidazole | 2-styryl...)
Affinity DataKi:  19nMAssay Description:Displacement of [125I]p-iodoclonidine from imidazoline receptor I-1 of PC12 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50138500(2-((E)-Styryl)-4,5-dihydro-1H-imidazole | 2-styryl...)
Affinity DataKi:  19nMAssay Description:Displacement of [125I]p-iodoclonidine from imidazoline receptor I-1 in rat pheochromocytoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50138500(2-((E)-Styryl)-4,5-dihydro-1H-imidazole | 2-styryl...)
Affinity DataKi:  3.80E+3nMAssay Description:Displacement of [125I]p-iodoclonidine from imidazoline receptor I-1 of PC12 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed