Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with Target = 'Nischarin' and Ligand = 'BDBM50179398'
TargetNischarin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50179398(CHEMBL94022)
Affinity DataKi:  11.7nMAssay Description:Displacement of [125I]p-iodoclonidine from imidazoline receptor I-1 of PC12 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50179398(CHEMBL94022)
Affinity DataKi:  12nMAssay Description:Displacement of [125I]p-iodoclonidine from imidazoline receptor I-1 of PC12 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)TBA
LigandPNGBDBM50179398(CHEMBL94022)
Affinity DataKi:  12nMAssay Description:Binding affinity to I1 imidazoline binding site in Rattus norvegicus (rat) PC12 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNischarin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50179398(CHEMBL94022)
Affinity DataKi:  12nMAssay Description:Displacement of [125I]p-iodoclonidine from imidazoline receptor I-1 in rat pheochromocytoma cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50179398(CHEMBL94022)
Affinity DataKi:  251nMAssay Description:Predicted affinity for imidazoline receptor I2 by three field CoMFA modelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(RAT)TBA
LigandPNGBDBM50179398(CHEMBL94022)
Affinity DataKi:  347nMAssay Description:Displacement of [125I]PIC from Imidazoline-1 receptor in rat PC12 cell membrane by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed