Affinity DataIC50: 200nMAssay Description:Inverse agonist activity at RORgammaT (unknown origin) by M1H assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.80E+4nMAssay Description:Inverse agonist activity at human RoRc-LBD fusion protein with GST expressed in BL-21 (BL3) cells assessed as SRC1 coactivator peptide recruitmentMore data for this Ligand-Target Pair