Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Nuclear receptor subfamily 1 group I member 2' and Ligand = 'BDBM50377913'
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50377913(HYPERFORIN)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]SR12813 from human PXR by scintillation proximity competition binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 1 group I member 2(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50377913(HYPERFORIN)
Affinity DataKi:  27nMAssay Description:Binding affinity to pregnane receptor in human hepatocytesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed