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Found 4 Enz. Inhib. hit(s) with Target = 'Orexin receptor type 2' and Ligand = 'BDBM163968'
TargetOrexin receptor type 2(Homo sapiens (Human))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM163968(US9062078, 99 | US9475819, 99 | US9637496, 99 | US...)
Affinity DataKi:  2.90E+3nM ΔG°:  -33.2kJ/moleT: 2°CAssay Description:HEK293 stably expressing human orexin 2 receptor (Genebank accession number NM001526) were grown to confluency in DMEM (Hyclone, cat #SH30022), 10% F...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOrexin receptor type 2(Homo sapiens (Human))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM163968(US9062078, 99 | US9475819, 99 | US9637496, 99 | US...)
Affinity DataKi:  2.90E+3nMAssay Description:HEK293 stably expressing human orexin 2 receptor (Genebank accession number NM_001526) were grown to confluency in DMEM (Hyclone, cat #SH30022), 10% ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOrexin receptor type 2(Homo sapiens (Human))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM163968(US9062078, 99 | US9475819, 99 | US9637496, 99 | US...)
Affinity DataKi:  2.90E+3nM ΔG°:  -33.2kJ/moleT: 2°CAssay Description:HEK293 stably expressing human orexin 2 receptor (Genebank accession number NM_001526) were grown to confluency in DMEM (Hyclone, cat # SH30022), 10%...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetOrexin receptor type 2(Homo sapiens (Human))
Janssen Pharmaceutica

US Patent
LigandPNGBDBM163968(US9062078, 99 | US9475819, 99 | US9637496, 99 | US...)
Affinity DataKi:  2.90E+3nM ΔG°:  -33.2kJ/moleT: 2°CAssay Description:HEK293 stably expressing human orexin 2 receptor (Genebank accession number NM_001526) were grown to confluency in DMEM (Hyclone, cat #SH30022), 10% ...More data for this Ligand-Target Pair
In DepthDetails US Patent