Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Oxysterols receptor LXR-alpha' and Ligand = 'BDBM50294738'
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50294738(CHEMBL551981 | {3-[3-Benzyl-8-(trifluoromethyl)qui...)
Affinity DataIC50:  1.12E+6nMAssay Description:Displacement of [3H]T0901317 from human recombinant N-terminal biotinylated tagged LXRalpha ligand binding domain (197-447) expressed in Escherichia ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50294738(CHEMBL551981 | {3-[3-Benzyl-8-(trifluoromethyl)qui...)
Affinity DataEC50:  1.35E+4nMAssay Description:Agonist activity at human LXRalpha ligand binding domain (205-448) expressed in human HuH7 cells cotransfected with Gal4-DBD by luciferase transactiv...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed