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Found 2 Enz. Inhib. hit(s) with Target = 'Oxytocin receptor' and Ligand = 'BDBM50271608'
TargetOxytocin receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50271608(CHEMBL4129142)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]OT from human mammary gland oxytocin receptor expressed in HEK293 cell membrane after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Imperial College

Curated by ChEMBL
LigandPNGBDBM50271608(CHEMBL4129142)
Affinity DataEC50:  34nMAssay Description:Agonist activity at human mammary gland oxytocin receptor expressed in CHO cells assessed as increase in intracellular calcium flux measured for 5 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed