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Found 1 Enz. Inhib. hit(s) with Target = 'P2X purinoceptor 7' and Ligand = 'BDBM50411429'
TargetP2X purinoceptor 7(Rattus norvegicus (Rat))
Astrazeneca R&D Charnwood

Curated by ChEMBL
LigandPNGBDBM50411429(CHEMBL235789)
Affinity DataIC50:  398nMAssay Description:Antagonist activity at rat P2X7 receptor transfected in HEK cells assessed as inhibition of benzylATP-induced changes in plasma membrane pore formati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed