Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with Target = 'P2Y purinoceptor 4' and Ligand = 'BDBM50118213'
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50118213(uridine 5'-(tetrahydrogen triphosphate) | UTP | 5'...)
Affinity DataEC50:  90nMAssay Description:Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate accumulation by scintillation proximity as...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50118213(uridine 5'-(tetrahydrogen triphosphate) | UTP | 5'...)
Affinity DataEC50:  550nMAssay Description:Agonist activity at human P2Y4 transfected in human 1321N1 cellsMore data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50118213(uridine 5'-(tetrahydrogen triphosphate) | UTP | 5'...)
Affinity DataEC50:  90nMAssay Description:Agonist activity at human recombinant P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate production by scintillation pr...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50118213(uridine 5'-(tetrahydrogen triphosphate) | UTP | 5'...)
Affinity DataEC50:  480nMAssay Description:Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by dual-excitatio...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50118213(uridine 5'-(tetrahydrogen triphosphate) | UTP | 5'...)
Affinity DataEC50:  39nMAssay Description:Agonist activity at human cloned P2Y4 receptor expressed in human 1321N1 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50118213(uridine 5'-(tetrahydrogen triphosphate) | UTP | 5'...)
Affinity DataEC50:  39nMAssay Description:Agonist activity at human cloned P2Y4 receptor expressed in human 1321N1 by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50118213(uridine 5'-(tetrahydrogen triphosphate) | UTP | 5'...)
Affinity DataEC50:  100nMAssay Description:Agonist activity evaluated as change in the level of cytosolic calcium in 1321N astrocytoma cells infected with a retrovirus encoding the human P2Y4 ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Rat)
National Institute of Diabetes

Curated by ChEMBL
LigandPNGBDBM50118213(uridine 5'-(tetrahydrogen triphosphate) | UTP | 5'...)
Affinity DataEC50:  2.60E+3nMAssay Description:The compound was evaluated for antagonist activity against phospholipase C coupled recombinant rat P2Y purinoceptor 4 (P2Y4)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50118213(uridine 5'-(tetrahydrogen triphosphate) | UTP | 5'...)
Affinity DataEC50:  2.50E+3nMAssay Description:The compound was evaluated for antagonist activity against phospholipase C coupled recombinant human P2Y purinoceptor 4 (P2Y4)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50118213(uridine 5'-(tetrahydrogen triphosphate) | UTP | 5'...)
Affinity DataEC50:  90nMAssay Description:Agonist activity at human P2Y4More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50118213(uridine 5'-(tetrahydrogen triphosphate) | UTP | 5'...)
Affinity DataEC50:  73nMAssay Description:Agonist activity at human recombinant P2Y4 receptor expressed in 1321N1 cells assessed as stimulation of phospholipase CMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50118213(uridine 5'-(tetrahydrogen triphosphate) | UTP | 5'...)
Affinity DataEC50:  87nMAssay Description:Agonist activity at human P2Y4 receptor expressed in 1321N1 cells assessed as IP accumulation by SPAMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50118213(uridine 5'-(tetrahydrogen triphosphate) | UTP | 5'...)
Affinity DataEC50:  500nMAssay Description:Agonist activity at human P2Y4 receptor expressed in human 1321N1 cells assessed as calcium elevation by fura2/AM assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50118213(uridine 5'-(tetrahydrogen triphosphate) | UTP | 5'...)
Affinity DataEC50:  900nMAssay Description:Agonist activity at human GFP-tagged P2Y4 receptor expressed in human 1321N1 cells assessed as intracellular calcium mobilization by fura2/AM-based f...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50118213(uridine 5'-(tetrahydrogen triphosphate) | UTP | 5'...)
Affinity DataEC50:  480nMAssay Description:Agonist activity at human P2Y purinoceptor 4 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrofl...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50118213(uridine 5'-(tetrahydrogen triphosphate) | UTP | 5'...)
Affinity DataEC50:  88nMAssay Description:Agonist activity at human recombinant P2Y4 receptor expressed in human 1321N1 cells assessed as [3H]inositol phosphate intracellular accumulation by ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetP2Y purinoceptor 4(Human)
Niddk

Curated by ChEMBL
LigandPNGBDBM50118213(uridine 5'-(tetrahydrogen triphosphate) | UTP | 5'...)
Affinity DataEC50:  80nMAssay Description:Agonist activity at human P2Y4More data for this Ligand-Target Pair
In DepthDetails Article
PubMed