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Found 2 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor alpha' and Ligand = 'BDBM50176609'
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50176609((R)-2-(3-((3-fluoro-4-(trifluoromethyl)benzamido)m...)
Affinity DataEC50:  150nMAssay Description:Transactivation of Gal4-fused human PPARalpha expressed in HEK293 cells after 16 to 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50176609((R)-2-(3-((3-fluoro-4-(trifluoromethyl)benzamido)m...)
Affinity DataEC50:  180nMAssay Description:Agonist activity at PPARalpha transfected in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed