Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor alpha' and Ligand = 'BDBM50235985'
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235985BDBM50235985(CHEMBL4092600)
Affinity DataKd:  0.75nMAssay Description:Binding affinity to PPARalpha (unknown origin) assessed as thermodynamic dissociation constant by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2019
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235985BDBM50235985(CHEMBL4092600)
Affinity DataEC50:  46nMAssay Description:Transactivation of GAL4-fused human PPARalpa LBD expressed in human HepG2 cells after 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2019
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor alpha(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50235985BDBM50235985(CHEMBL4092600)
Affinity DataKon:  0.0160M-1s-1Assay Description:Binding affinity to PPARalpha (unknown origin) assessed as kinetic dissociation constant by SPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/12/2019
Entry Details Article
PubMed