Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor alpha' and Ligand = 'BDBM50275922'
LigandChemical structure of BindingDB Monomer ID 50275922BDBM50275922((S)-2-(4-chlorophenoxy)-3-(4-phenoxyphenyl)propano...)
Affinity DataEC50:  27nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells co-transfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50275922BDBM50275922((S)-2-(4-chlorophenoxy)-3-(4-phenoxyphenyl)propano...)
Affinity DataEC50:  900nMAssay Description:Agonist activity at GAL4-fused PPARalpha A454M mutant (unknown origin) expressed in human HepG2 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50275922BDBM50275922((S)-2-(4-chlorophenoxy)-3-(4-phenoxyphenyl)propano...)
Affinity DataEC50:  3.90E+3nMAssay Description:Agonist activity at GAL4-fused PPARalpha (unknown origin) expressed in human HepG2 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
LigandChemical structure of BindingDB Monomer ID 50275922BDBM50275922((S)-2-(4-chlorophenoxy)-3-(4-phenoxyphenyl)propano...)
Affinity DataEC50:  3.90E+3nMAssay Description:Agonist activity at GAL4-fused PPARalpha (unknown origin) expressed in human HepG2 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed