Found 3 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor delta' and Ligand = 'BDBM50214207'
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Tokyo
Curated by ChEMBL
University Of Tokyo
Curated by ChEMBL
Affinity DataEC50: 0.910nMAssay Description:Effect on PPARdelta transactivation activity in HEK293 cellsMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Tokyo
Curated by ChEMBL
University Of Tokyo
Curated by ChEMBL
Affinity DataEC50: 0.720nMAssay Description:Transactivation of Gal4-fused human PPARdelta expressed in HEK293 cells after 16 to 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Tokyo
Curated by ChEMBL
University Of Tokyo
Curated by ChEMBL
Affinity DataEC50: 0.720nMAssay Description:Agonist activity at PPARdelta receptor expressed in HEK293 cells cotransfected with GAL4 by transactivation assayMore data for this Ligand-Target Pair