Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor delta' and Ligand = 'BDBM50214209'
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50214209((R)-2-(4-butoxy-3-((2-fluoro-4-(trifluoromethyl)be...)
Affinity DataEC50:  8.5nMAssay Description:Transactivation of Gal4-fused human PPARdelta expressed in HEK293 cells after 16 to 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Okayama University

Curated by ChEMBL
LigandPNGBDBM50214209((R)-2-(4-butoxy-3-((2-fluoro-4-(trifluoromethyl)be...)
Affinity DataEC50:  8.30nMAssay Description:Effect on PPARdelta transactivation activity in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed