Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor gamma' and Ligand = 'BDBM50171897'
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50171897((S)-2-(4-chlorophenoxy)-3-phenylpropanoic acid | (...)
Affinity DataEC50:  2.69E+3nMAssay Description:Agonist activity at GAL4-fused PPARgamma (unknown origin) expressed in human HepG2 cells by transactivation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50171897((S)-2-(4-chlorophenoxy)-3-phenylpropanoic acid | (...)
Affinity DataEC50:  2.70E+3nMAssay Description:Effective concentration against human PPARgamma expressed in HepG2 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50171897((S)-2-(4-chlorophenoxy)-3-phenylpropanoic acid | (...)
Affinity DataEC50:  7.94E+3nMAssay Description:Agonist activity at human PPARgamma ligand binding domain expressed in human HepG2 cells co-transfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetPeroxisome proliferator-activated receptor gamma(Human)
University of Bari Aldo Moro

Curated by ChEMBL
LigandPNGBDBM50171897((S)-2-(4-chlorophenoxy)-3-phenylpropanoic acid | (...)
Affinity DataEC50:  9.60E+3nMAssay Description:Agonist activity at GAL4-tagged human PPARgamma ligand binding domain expressed in HepG2 cells assessed as transactivation after 20 hrs by beta-galac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed