Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor gamma' and Ligand = 'BDBM50322683'
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50322683(4-Anilino-6-(benzylthio)-2-(methylthio)pyrimidine-...)
Affinity DataEC50:  1.60E+3nMAssay Description:Partial agonist activity at human PPARgamma-LBD expressed in CHO-K1 cells co-transfected with GAL4 assessed as luciferase activity by transactivation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed