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Found 1 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor gamma' and Ligand = 'BDBM50322686'
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Kyorin Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50322686(4-(Benzylthio)-2-(methylthio)-6-(3-pyridylmethylam...)
Affinity DataEC50:  740nMAssay Description:Partial agonist activity at human PPARgamma-LBD expressed in CHO-K1 cells co-transfected with GAL4 assessed as luciferase activity by transactivation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed