Found 6 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor gamma' and Ligand = 'BDBM50322695' TargetPeroxisome proliferator-activated receptor gamma(Rattus norvegicus)
Kyorin Pharmaceutical Co., Ltd
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 539nMAssay Description:Antagonist activity at rat PPARgamma-LBD expressed in CHO-K1 cells co-transfected with GAL4 assessed as inhibition of rosiglitazone-induced luciferas...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Kyorin Pharmaceutical Co., Ltd
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 1.77E+3nMAssay Description:Antagonist activity at mouse PPARgamma-LBD expressed in CHO-K1 cells co-transfected with GAL4 assessed as inhibition of rosiglitazone-induced lucifer...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Kyorin Pharmaceutical Co., Ltd
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataIC50: 1.79E+3nMAssay Description:Antagonist activity at human PPARgamma-LBD expressed in CHO-K1 cells co-transfected with GAL4 assessed as inhibition of rosiglitazone-induced lucifer...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Mus musculus)
Kyorin Pharmaceutical Co., Ltd
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataEC50: 158nMAssay Description:Partial agonist activity at mouse PPARgamma-LBD expressed in CHO-K1 cells co-transfected with GAL4 assessed as luciferase activity by transactivation...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Kyorin Pharmaceutical Co., Ltd
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataEC50: 140nMAssay Description:Partial agonist activity at human PPARgamma-LBD expressed in CHO-K1 cells co-transfected with GAL4 assessed as luciferase activity by transactivation...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Rattus norvegicus)
Kyorin Pharmaceutical Co., Ltd
Curated by ChEMBL
Kyorin Pharmaceutical Co., Ltd
Curated by ChEMBL
Affinity DataEC50: 158nMAssay Description:Partial agonist activity at rat PPARgamma-LBD expressed in CHO-K1 cells co-transfected with GAL4 assessed as luciferase activity by transactivation a...More data for this Ligand-Target Pair
