
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Goethe-University
Curated by ChEMBL
Goethe-University
Curated by ChEMBL
Affinity DataIC50: 650nMAssay Description:Partial agonist activity at recombinant sGSF-PPARgamma (unknown origin) assessed as reduction in rosiglitazone induced CBP-1 recruitment incubated fo...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Goethe-University
Curated by ChEMBL
Goethe-University
Curated by ChEMBL
Affinity DataEC50: 150nMAssay Description:Partial agonist activity at GAL4-tagged human PPARgamma LBD expressed in HEK293T cells incubated for 12 to 14 hrs by dual-Glo luciferase assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Goethe-University
Curated by ChEMBL
Goethe-University
Curated by ChEMBL
Affinity DataEC50: 180nMAssay Description:Partial agonist activity at sGSF-PPARgamma (unknown origin) assessed as CBP-1 recruitment by HT-FRET assayMore data for this Ligand-Target Pair
