Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Pituitary adenylate cyclase-activating polypeptide type I receptor' and Ligand = 'BDBM50250087'
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250087(CHEMBL499665 | [Aib4]PACAP38)
Affinity DataIC50:  9.20nMAssay Description:Displacement of [125I]Ac-PACAP27 from human recombinant PAC1 receptor expressed in CHO cells by gamma- counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPituitary adenylate cyclase-activating polypeptide type I receptor(Homo sapiens (Human))
Institut National De La Recherche Scientifique

Curated by ChEMBL
LigandPNGBDBM50250087(CHEMBL499665 | [Aib4]PACAP38)
Affinity DataEC50:  3.30nMAssay Description:Agonist activity at human recombinant PAC1 receptor expressed in CHO cells assessed as PACAP38-induced calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed