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Report error Found 4 Enz. Inhib. hit(s) with Target = 'Platelet-derived growth factor receptor alpha/beta' and Ligand = 'BDBM50534293'
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50534293(CHEMBL3341966)
Affinity DataIC50: 110nMAssay Description:Partial agonist activity at alpha4beta2 nAChR in HEK293 cells assessed as reduction in Ca+2 influx by FLIPR assyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50534293(CHEMBL3341966)
Affinity DataIC50: 260nMAssay Description:Partial agonist activity at alpha3beta4 nAChR in HEK293 cells assessed as reduction in Ca+2 influx by FLIPR assyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50534293(CHEMBL3341966)
Affinity DataKi:  21nMAssay Description:Displacement of [3H] epibatidine from alpha3beta4 nAChR in HEK293 cells assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
TargetPlatelet-derived growth factor receptor alpha/beta(Mouse)
University of Illinois At Chicago

Curated by ChEMBL
LigandPNGBDBM50534293(CHEMBL3341966)
Affinity DataKi:  21nMAssay Description:Displacement of [3H] epibatidine from alpha4beta2 nAChR in HEK293 cells assessed as inhibition constantMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed