Report error Found 46 Enz. Inhib. hit(s) with Target = 'Progesterone receptor' and Ligand = 'BDBM8903'
Affinity DataKi: 3.40nMAssay Description:Binding affinity at human progesterone receptorMore data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataKi: 3.5nMAssay Description:Displacement of [3H]progesterone from Progesterone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Binding affinity determined for human Progesterone receptor A isoformMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:The binding affinity measured using baculovirus-expressed hPR-A in sf21 cells.More data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Binding affinity against baculovirus expressed human Progesterone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Binding affinity was determined against hPR-A (human progesterone receptor) using progesterone radioligand in competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Binding affinity against human progesterone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Binding affinity to human progesterone receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Binding affinity towards human progesterone receptor A isoform using progesterone as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Human progesterone receptor (hPR) agonist activity in T47D human breast cancer cell lineMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:The binding affinity of the compound was determined on Human progesterone receptor (hPR-A) using progesterone as radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Binding affinity for human progesterone receptor isoform A expressed in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Displacement of [3H]progesterone from human progesterone receptor B after 16 hrs by scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 10.4nMAssay Description:Inhibition of [3H]-R5020 binding to rabbit uterine progesterone receptorChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Binding affinity to progesterone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60nMT: 22°CAssay Description:Competitive binding assay were performed using increasing dose of the contrast agents and fluorescently labeled progesterone as the competitor. More data for this Ligand-Target Pair
Affinity DataIC50: 3.5nMAssay Description:Binding affinity for Progesterone receptor (PR) in human T47D breast carcinoma cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Binding affinity towards human progesterone receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Displacement of [3H]progesterone from rabbit PR by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Displacement of [3H]progesterone from progesterone receptor in JW rabbit uterus after 2 hrs by liquid scintillation countingChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Binding affinity against Progesterone receptor in human TE85 osteosarcoma cells was determined using (Z)-[125I]-17-alpha-(2-iodovinyl)-19-nor-testost...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human progesterone receptor B expressed in african green monkey CV1 cells co-transfected with MMTV-Luc assessed as effect on p...More data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Agonist activity at human PRMore data for this Ligand-Target Pair
Affinity DataEC50: 0.920nMAssay Description:Effective concentration against PR (progesterone receptor)More data for this Ligand-Target Pair
Affinity DataEC50: 15.2nMAssay Description:Agonist activity at human progesterone receptor B expressed in african green monkey CV1 cells co-transfected with MMTV-Luc after 24 hrs by luciferase...More data for this Ligand-Target Pair
Affinity DataEC50: 2.90nMAssay Description:Effective concentration for agonist activity towards human progesterone receptor (hPR) using the cotransfection assay in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.90nMAssay Description:Human progesterone receptor (hPR) agonist activity in T47D human breast cancer cell lineMore data for this Ligand-Target Pair
Affinity DataEC50: 0.900nMAssay Description:Effective concentration on alkaline phosphatase activity in human T47D breast carcinoma cell line.More data for this Ligand-Target Pair
Affinity DataEC50: 0.900nMAssay Description:Activity at progesterone receptor assessed as alkaline phosphatase activity in human T47D cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.100nMAssay Description:Activation of progesterone receptor in human T47D cells after 20 hrs by PRE-tagged luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.90nMAssay Description:Compound was tested for agonistic activity by cotransfection assay against human Progesterone receptor in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.80nMAssay Description:Agonistic activity by cotransfection assay against human Progesterone receptor in T47D cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.20nMAssay Description:Agonist activity at human progesterone receptor in human T47D cells assessed as alkaline phosphatase activityMore data for this Ligand-Target Pair
Affinity DataEC50: 0.5nMAssay Description:Agonist activity at human progesterone receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 2nMAssay Description:Agonist activity at human PRGR expressed in HEK293 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 2.90nMAssay Description:Agonistic activity against human progesterone receptor in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.80nMAssay Description:Agonistic activity against human progesterone receptor in T47D breast cancer cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.90nMAssay Description:Agonist activity was determined against hPR (human progesterone receptor) compared to that of progesterone (100%)More data for this Ligand-Target Pair
Affinity DataEC50: 2.90nMAssay Description:Effective concentration (EC50) against human progesterone receptor expressed in CV-1 cellMore data for this Ligand-Target Pair
Affinity DataEC50: 1.5nMAssay Description:Effective concentration for half-maximal activation of human progesterone receptor expressed in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.90nMAssay Description:Agonistic activity was measured for modulation of hPR-B (human progesterone receptor) in co-transfected CV-1 cells.More data for this Ligand-Target Pair
Affinity DataEC50: 2.90nMAssay Description:Agonistic activity to the human progesterone receptor(hPR)assayed in CV-1 cells in cotransfection assay.More data for this Ligand-Target Pair
Affinity DataEC50: 0.920nMAssay Description:Agonistic activity against progesterone receptor in alkaline phosphatase assay using human T47D breast carcinoma cell lineMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Antagonist activity against hPR (human progesterone receptor) compared to that of progesterone (100%)More data for this Ligand-Target Pair
Affinity DataEC50: 0.180nMAssay Description:Agonist activity at PR in human T47D cells using p-nitrophenyl phosphate as substrate assessed as induction of alkaline phosphatase activity incubate...More data for this Ligand-Target Pair
Affinity DataEC50: 1.80nMAssay Description:Human progesterone receptor (hPR) agonist activity in T47D human breast cancer cell lineMore data for this Ligand-Target Pair
