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Found 4 Enz. Inhib. hit(s) with Target = 'Prostaglandin D2 receptor' and Ligand = 'BDBM50060448'
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060448((+) 7-[3-(2-Phenyl-1H-indole-6-sulfonylamino)-bicy...)
Affinity DataIC50:  47nMAssay Description:Inhibition of [3H]-PGD-2 specific binding to Prostaglandin D2 receptor fromhuman platelet membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060448((+) 7-[3-(2-Phenyl-1H-indole-6-sulfonylamino)-bicy...)
Affinity DataIC50:  47nMAssay Description:In vitro inhibition of [3H]- PGD-2 radioligand binding to prostaglandin D2 receptor on human platelet membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060448((+) 7-[3-(2-Phenyl-1H-indole-6-sulfonylamino)-bicy...)
Affinity DataIC50:  71nMAssay Description:In vitro inhibition of cAMP formation evoked by prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50060448((+) 7-[3-(2-Phenyl-1H-indole-6-sulfonylamino)-bicy...)
Affinity DataIC50:  120nMAssay Description:Inhibition of cAMP formation evoked by the prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed