Affinity DataKi: 1.10nMAssay Description:Binding affinity to human DP receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.290nMAssay Description:Activity at human DP receptor in washed platelets assessed as inhibition of PGD2-induced cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Activity at human DP receptor in platelet rich plasma assessed as inhibition of PGD2-induced cAMP accumulationMore data for this Ligand-Target Pair