Found 4 Enz. Inhib. hit(s) with Target = 'Prostaglandin E2 receptor EP1 subtype' and Ligand = 'BDBM50160917'
Affinity DataKi: 0.300nMAssay Description:Antagonist activity against PGE2 activated EP1 receptor assessed as ability to inhibit intracellular calcium mobilisation by FLIPRMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Binding affinity against Prostaglandin E receptor was determined in humanMore data for this Ligand-Target Pair
Affinity DataKi: 70nMAssay Description:Binding affinity against Prostaglandin E receptor in presence of 2% human serum albuminMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Displacement of [3H]PGE2 from human EP1 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair