Found 6 Enz. Inhib. hit(s) with Target = 'Prostaglandin E2 receptor EP2 subtype' and Ligand = 'BDBM50156547'
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Emd-Serono Research Institute
Curated by ChEMBL
Emd-Serono Research Institute
Curated by ChEMBL
Affinity DataKi: 120nMAssay Description:Displacement of [3H]PGE2 from human EP2 receptorMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Emd-Serono Research Institute
Curated by ChEMBL
Emd-Serono Research Institute
Curated by ChEMBL
Affinity DataKi: 130nMAssay Description:Binding affinity to human EP2 receptorMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP2 subtype(Mus musculus (Mouse))
Minase Research Institute
Curated by ChEMBL
Minase Research Institute
Curated by ChEMBL
Affinity DataKi: 340nMAssay Description:Displacement of [3H]-PGE2 from mouse EP2 receptor expressed in CHO cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP2 subtype(Mus musculus (Mouse))
Minase Research Institute
Curated by ChEMBL
Minase Research Institute
Curated by ChEMBL
Affinity DataKi: >340nMAssay Description:Displacement of [3H]-PGE2 from mouse EP2 receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP2 subtype(Homo sapiens (Human))
Emd-Serono Research Institute
Curated by ChEMBL
Emd-Serono Research Institute
Curated by ChEMBL
Affinity DataEC50: 15nMAssay Description:Agonist activity at human EP2 receptor by cAMP assayMore data for this Ligand-Target Pair
TargetProstaglandin E2 receptor EP2 subtype(Rattus norvegicus)
Minase Research Institute
Curated by ChEMBL
Minase Research Institute
Curated by ChEMBL
Affinity DataEC50: 1.80E+3nMAssay Description:Agonist activity at rat EP2 receptorMore data for this Ligand-Target Pair