Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with Target = 'Prostaglandin E2 receptor EP3 subtype' and Ligand = 'BDBM50307409'
TargetProstaglandin E2 receptor EP3 subtype(Mouse)
Minase Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50307409BDBM50307409(3-(2-(3-methyl-1-phenylbutylcarbamoyl)-4-(phenoxym...)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]PGE2 from mouse EP3 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Mouse)
Minase Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50307409BDBM50307409(3-(2-(3-methyl-1-phenylbutylcarbamoyl)-4-(phenoxym...)
Affinity DataKi:  0.700nMAssay Description:Displacement of [3H]PGE3alpha from mouse EP3alpha receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Mouse)
Minase Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50307409BDBM50307409(3-(2-(3-methyl-1-phenylbutylcarbamoyl)-4-(phenoxym...)
Affinity DataIC50: 68nMAssay Description:Antagonist activity at mouse EP3alpha receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase in intracellular calcium level ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2010
Entry Details Article
PubMed
TargetProstaglandin E2 receptor EP3 subtype(Mouse)
Minase Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50307409BDBM50307409(3-(2-(3-methyl-1-phenylbutylcarbamoyl)-4-(phenoxym...)
Affinity DataIC50: 68nMAssay Description:Antagonist activity at mouse EP3 receptor expressed in CHO cells assessed as inhibition of PGE2-induced increase intracellular calcium level in prese...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/1/2010
Entry Details Article
PubMed