Found 50 Enz. Inhib. hit(s) with Target = 'Prostaglandin G/H synthase 1' and Ligand = 'BDBM22360' TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
St. Bartholomew'S And The Royal London School Of Medicine And Dentistry
Curated by PDSP Ki Database
St. Bartholomew'S And The Royal London School Of Medicine And Dentistry
Curated by PDSP Ki Database
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
St. Bartholomew'S And The Royal London School Of Medicine And Dentistry
Curated by PDSP Ki Database
St. Bartholomew'S And The Royal London School Of Medicine And Dentistry
Curated by PDSP Ki Database
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
St. Bartholomew'S And The Royal London School Of Medicine And Dentistry
Curated by PDSP Ki Database
St. Bartholomew'S And The Royal London School Of Medicine And Dentistry
Curated by PDSP Ki Database
Affinity DataKi: 6.20E+4nMAssay Description:Inhibition of COX-1 (unknown origin) using arachidonic acid as substrate assessed as formation of prostanoid products preincubated for 10 mins prior ...More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of ovine COX1 by enzyme immunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of ovine COX1 by enzyme immunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of ovine COX1More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of ovine COX1 by enzyme immuno assayMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of sheep COX1 by enzyme immunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of Ovine COX-1 assessed as decrease in prostaglandin production using arachidonic acid as substrate pretreated for 15 mins followed by sub...More data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of ovine COX-1 assessed as reduction in PGF2-alpha formation using arachidonic acid as substrate by enzyme immunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of ovine COX1 by enzyme immunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of ovine COX1 by enzyme immuno assayMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of ovine COX1 by enzyme immuno assayMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:In vitro inhibitory concentration of the compound against COX-1 enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:Inhibition of ovine COX1 by enzyme immuno assayMore data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:Inhibition of bovine COX-1 by enzyme immuno assayMore data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:Inhibition of ovine COX1More data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:Inhibition of ovine COX1 by enzyme immunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:Inhibition of ovine COX-1 by enzyme immuno assayMore data for this Ligand-Target Pair
Affinity DataIC50: 350nMpH: 8.0 T: 2°CAssay Description:The COX enzyme activities were measured using the COX Inhibitor Screening Assay kit provided by Cayman (Cayman, Chemical Co., Ann Arbor, MI). The as...More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
St. Bartholomew'S And The Royal London School Of Medicine And Dentistry
Curated by PDSP Ki Database
St. Bartholomew'S And The Royal London School Of Medicine And Dentistry
Curated by PDSP Ki Database
Affinity DataIC50: 350nMAssay Description:Inhibition of COX1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:Inhibition of ovine COX1 by enzyme immuno assayMore data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:Inhibition of ovine COX1More data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:Inhibition of ovine COX1 by enzyme immuno assayMore data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:Inhibition of ovine COX1 by enzyme immuno assayMore data for this Ligand-Target Pair
Affinity DataIC50: 350nMAssay Description:In vitro inhibition of ovine prostaglandin G/H synthase 1More data for this Ligand-Target Pair
Affinity DataIC50: 411nMAssay Description:Inhibition of ovine COX-1 assessed as inhibition of transformation of AA to PGH2 by EIAMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:The ability of the test compounds to inhibit ovine COX01 and human recombinant COX-2 was determined using an enzyme immuno assay (EIA) kit according ...More data for this Ligand-Target Pair
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of sheep COX1-mediated PGE2 production after 2 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 6.12E+3nMAssay Description:Inhibition of ovine COX1 using arachidonic acid as substrate pretreated for 5 mins followed by substrate addition and measured after 2 mins by fluore...More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Ovine COX-1 preincubated for 15 mins by fluorescence analysisMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
St. Bartholomew'S And The Royal London School Of Medicine And Dentistry
Curated by PDSP Ki Database
St. Bartholomew'S And The Royal London School Of Medicine And Dentistry
Curated by PDSP Ki Database
Affinity DataIC50: 1.14E+4nMAssay Description:Inhibition of COX1 by radioimmunoassay methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibitory concentration in DMSO with purified ovine Prostaglandin G/H synthase 1 (COX-1).More data for this Ligand-Target Pair
Affinity DataIC50: 9.00E+4nMAssay Description:Inhibition of ovine COX1 by measuring PGE2More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
St. Bartholomew'S And The Royal London School Of Medicine And Dentistry
Curated by PDSP Ki Database
St. Bartholomew'S And The Royal London School Of Medicine And Dentistry
Curated by PDSP Ki Database
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of COX1More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
St. Bartholomew'S And The Royal London School Of Medicine And Dentistry
Curated by PDSP Ki Database
St. Bartholomew'S And The Royal London School Of Medicine And Dentistry
Curated by PDSP Ki Database
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of COX1More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of ovine COX1More data for this Ligand-Target Pair
Affinity DataIC50: 2.40E+5nMAssay Description:Inhibitory activity against Prostaglandin G/H synthase 1 isolated from ram (sheep) seminal vesicleMore data for this Ligand-Target Pair
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of ovine COX1More data for this Ligand-Target Pair
Affinity DataIC50: 3.42E+5nMAssay Description:Inhibition of bovine seminal microsomal COX1 assessed as PGE2 production preincubated for 10 minsMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
St. Bartholomew'S And The Royal London School Of Medicine And Dentistry
Curated by PDSP Ki Database
St. Bartholomew'S And The Royal London School Of Medicine And Dentistry
Curated by PDSP Ki Database
Affinity DataIC50: 5.60E+5nMAssay Description:Inhibition of COX1 after 5 mins by spectrophotometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 6.00E+5nMAssay Description:Antagonistic potency for NK-1 receptor was determined in a radioligand binding assay using IM9 human lymphoblastoma cell line.More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
St. Bartholomew'S And The Royal London School Of Medicine And Dentistry
Curated by PDSP Ki Database
St. Bartholomew'S And The Royal London School Of Medicine And Dentistry
Curated by PDSP Ki Database
Affinity DataIC50: 7.50E+5nMAssay Description:Inhibition of COX1More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
St. Bartholomew'S And The Royal London School Of Medicine And Dentistry
Curated by PDSP Ki Database
St. Bartholomew'S And The Royal London School Of Medicine And Dentistry
Curated by PDSP Ki Database
Affinity DataIC50: 7.80E+5nMAssay Description:Inhibition of COX1 by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibition of bovine seminal vesicle microsomal COX1-mediated prostaglandin productionMore data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Homo sapiens (Human))
St. Bartholomew'S And The Royal London School Of Medicine And Dentistry
Curated by PDSP Ki Database
St. Bartholomew'S And The Royal London School Of Medicine And Dentistry
Curated by PDSP Ki Database
Affinity DataIC50: 1.05E+6nMAssay Description:Inhibition of PGHS1 assessed as conversion of arachidonic acid to prostaglandinMore data for this Ligand-Target Pair
Affinity DataIC50: 1.28E+6nMAssay Description:Tested for inhibitory activity against Prostaglandin G/H synthase 1 from ovineMore data for this Ligand-Target Pair
Affinity DataIC50: 3.77E+6nMAssay Description:Inhibition of bovine seminal microsomal COX1 assessed as PGE2 productionMore data for this Ligand-Target Pair
Affinity DataIC50: 1.88E+7nMAssay Description:Inhibition of COX1 from ram seminal vesicles by liquid scintillation counterMore data for this Ligand-Target Pair
Affinity DataIC50: 4.97E+7nMAssay Description:Inhibition of sheep placental COX2 by liquid scintillation counterMore data for this Ligand-Target Pair
